A small molecule inhibitor of β-catenin/cyclic AMP response element-binding protein transcription KH Emami, C Nguyen, H Ma, DH Kim, KW Jeong, M Eguchi, RT Moon, ... Proceedings of the National Academy of Sciences 101 (34), 12682-12687, 2004 | 998 | 2004 |
Recent advances in selective opioid receptor agonists and antagonists M Eguchi Medicinal research reviews 24 (2), 182-212, 2004 | 216 | 2004 |
Chemogenomic identification of Ref-1/AP-1 as a therapeutic target for asthma C Nguyen, JL Teo, A Matsuda, M Eguchi, EY Chi, WR Henderson Jr, ... Proceedings of the National Academy of Sciences 100 (3), 1169-1173, 2003 | 129 | 2003 |
ICG-001, A Novel Small Molecule Regulator of TCF/β-Catenin Masakatsu Transcription M Eguchi, C Nguyen, SC Lee, M Kahn Medicinal chemistry 1 (5), 467-472, 2005 | 121 | 2005 |
Design, synthesis, and evaluation of opioid analogues with non-peptidic β-turn scaffold: enkephalin and endomorphin mimetics M Eguchi, RYW Shen, JP Shea, MS Lee, M Kahn Journal of medicinal chemistry 45 (7), 1395-1398, 2002 | 120 | 2002 |
New and efficient route to pipecolic acid derivatives by means of Rh-catalyzed intramolecular cyclohydrocarbonylation I Ojima, M Tzamarioudaki, M Eguchi The Journal of Organic Chemistry 60 (22), 7078-7079, 1995 | 105 | 1995 |
Enantioselective conjugate addition to cyclic enones with scalemic lithium organo (amido) cuprates, Part IV. Relationship between ligand structure and enantioselectivity BE Rossiter, M Eguchi, G Miao, NM Swingle, AE Hernández, D Vickers, ... Tetrahedron 49 (5), 965-986, 1993 | 103 | 1993 |
Solid-Phase Synthesis and Structural Analysis of Bicyclic β-Turn Mimetics Incorporating Functionality at the i to i + 3 Positions M Eguchi, MS Lee, H Nakanishi, M Stasiak, S Lovell, M Kahn Journal of the American Chemical Society 121 (51), 12204-12205, 1999 | 102 | 1999 |
Secondary structure peptide mimetics: Design, synthesis, and evaluation of β-strand mimetic thrombin inhibitors PD Boatman, CO Ogbu, M Eguchi, HO Kim, H Nakanishi, B Cao, JP Shea, ... Journal of medicinal chemistry 42 (8), 1367-1375, 1999 | 98 | 1999 |
Design, synthesis, and application of peptide secondary structure mimetics. M Eguchi, M Kahn Mini reviews in medicinal chemistry 2 (5), 447-462, 2002 | 76 | 2002 |
Silylformylation catalyzed by Rh and Rh-Co mixed metal complexes and its application to the synthesis of pyrrolizidine alkaloids I Ojima, RJ Donovan, M Eguchi, WR Shay, P Ingallina, A Korda, Q Zeng Tetrahedron 49 (25), 5431-5444, 1993 | 70 | 1993 |
Synthesis of pyrrolizidine alkaloids via rhodium-catalyzed silylformylation and amidocarbonylation M Eguchi, Q Zeng, A Korda, I Ojima Tetrahedron letters 34 (6), 915-918, 1993 | 66 | 1993 |
Enantioselective conjugate addition with chiral amidocuprates BE Rossiter, M Eguchi Tetrahedron letters 31 (7), 965-968, 1990 | 54 | 1990 |
Reverse-turn mimetics and methods relating thereto M Kahn, M Eguchi, HO Kim US Patent 6,013,458, 2000 | 52 | 2000 |
Solid-phase synthesis and solution structure of bicyclic β-turn peptidomimetics: diversity at the i position M Eguchi, MS Lee, M Stasiak, M Kahn Tetrahedron Letters 42 (7), 1237-1239, 2001 | 47 | 2001 |
Enantioselective conjugate addition to cyclic enones with (S)-mapp-cuprates. BE Rossiter, M Eguchi, AE Herna, D Vickers, J Medich, J Marr, D Heinis Tetrahedron letters 32 (32), 3973-3976, 1991 | 45 | 1991 |
Sam68 allows selective targeting of human cancer stem cells YD Benoit, RR Mitchell, RM Risueño, L Orlando, B Tanasijevic, AL Boyd, ... Cell Chemical Biology 24 (7), 833-844. e9, 2017 | 44 | 2017 |
Reverse-turn mimetics and methods relating thereto M Kahn, M Eguchi, HO Kim, M Stasiak US Patent 6,184,223, 2001 | 40 | 2001 |
β-sheet mimetics and use thereof as inhibitors of biologically active peptides or proteins M Kahn, CO Ogbu, M Eguchi, HO Kim, PD Boatman Jr US Patent 6,245,764, 2001 | 34 | 2001 |
Comprehensive Organometallic Chemistry II I Ojima, M Eguchi, M Tzamarioudaki, ... by EW Abel, FGA Stone, G. Wilkinson, and LS Hegedous, Pergamon, Oxford 12, 9-39, 1995 | 34 | 1995 |